1. Signaling Pathways
  2. Membrane Transporter/Ion Channel
  3. Na+/K+ ATPase
  4. Na+/K+ ATPase Antagonist

Na+/K+ ATPase Antagonist

Na+/K+ ATPase Antagonist (1):

Cat. No. Product Name Effect Purity
  • HY-12283
    Rostafuroxin
    Antagonist 98.00%
    Rostafuroxin (PST 2238), a digitoxigenin derivative, is an orally active and potent Na+,K+-ATPase (ATP1A1) antognist. Rostafuroxin binds specifically to the ATP1A1 extracellular domain and blocks respiratory syncytial virus (RSV)-triggered EGFR Tyr845 phosphorylation. Rostafuroxin has antihypertensive and anti-RSV activity.